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N-desmethyl Enzalutamide

CAS No. 1242137-16-1

N-desmethyl Enzalutamide ( N-desmethyl MDV3100;N-desmethyl MDV 3100;N-desmethyl MDV-3100 )

Catalog No. M10977 CAS No. 1242137-16-1

Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 43 Get Quote
5MG 72 Get Quote
10MG 102 Get Quote
25MG 210 Get Quote
50MG 404 Get Quote
100MG 593 Get Quote
500MG 1251 Get Quote
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Biological Information

  • Product Name
    N-desmethyl Enzalutamide
  • Note
    Research use only, not for human use.
  • Brief Description
    Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.
  • Description
    Amajor metabolite of Enzalutamide (MDV3100) which is an androgen-receptor (AR) antagonist for treatment of prostate cancer.
  • Synonyms
    N-desmethyl MDV3100;N-desmethyl MDV 3100;N-desmethyl MDV-3100
  • Pathway
    Endocrinology/Hormones
  • Target
    Androgen Receptor (AR)
  • Recptor
    Androgen Receptor (AR)
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1242137-16-1
  • Formula Weight
    450.41
  • Molecular Formula
    C20H14F4N4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 48 mg/mL
  • SMILES
    CC1(C(=O)N(C(=S)N1C2=CC(=C(C=C2)C(=O)N)F)C3=CC(=C(C=C3)C#N)C(F)(F)F)C
  • Chemical Name
    Benzamide, 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-thioxo-1-imidazolidinyl]-2-fluoro-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Tran C, et al. Science. 2009 May 8;324(5928):787-90.
2. Richards J, et al. Cancer Res. 2012 May 1;72(9):2176-82.
3. Gibbons JA, et al. Clin Pharmacokinet. 2015 Oct;54(10):1043-55.
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